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SGK1-IN-1 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5753902

MBS5753902 is an inhibitor targeting SGK1-IN-1. SGK1-IN-1 is a highly active and selective SGK-1 inhibitor(IC50 of 1nM). More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
SGK1-IN-1, Inhibitor
Full Product Name
SGK1-IN-1
Product Gene Name
SGK1-IN-1, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
418.83
Solubility
<1mg/ml refers to the product slightly soluble or insoluble
Formula
C17H12ClFN6O2S
SMILES
O=S(C1=C(F)C=CC(Cl)=C1)(NC2=CC=C(C3=NC(NN=C4N)=C4N=C3)C=C2)=O
CAS Number
1279829-87-6
Target & IC50
SGK-1: ic50 1nM

Structure of SGK1-IN-1, inhibitor

SGK1-IN-1 Inhibitor – Cat# MBS5753902

Product References and Citations for SGK1-IN-1, inhibitor

ARYL SULFONOHYDRAZIDES. WO 2013041119 A1.
ARYL SULFONOHYDRAZIDES. WO 2013041119 A1.
Halland N, et al. Discovery of N-[4-(1H-Pyrazolo[3,4-b]pyrazin-6-yl)-phenyl]-sulfonamides as Highly Active and Selective SGK1 Inhibitors. ACS Med Chem Lett. 2014 Oct 23;6(1):73-8.
Halland N, et al. Discovery of N-[4-(1H-Pyrazolo[3,4-b]pyrazin-6-yl)-phenyl]-sulfonamides as Highly Active and Selective SGK1 Inhibitors. ACS Med Chem Lett. 2014 Oct 23;6(1):73-8.

Other Notes

Small volumes of SGK1-IN-1, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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