Taltirelin acetate Inhibitor

Name: Taltirelin acetate Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5753999
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5753999

Taltirelin acetate is a superagonist at thyrotropin-releasing hormone receptor (TRH-R)(IC50 of 910nM and EC50 of 36nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release)). More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Taltirelin acetate, Inhibitor

Full Product Name

Taltirelin acetate

Product Synonym Names

TA-0910 acetate

Form/Format

Solid. Powder

Purity/Purification

99.44%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

465.46

Solubility

DMSO: 125mg/mL (268.55mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)

Formula

C19H27N7O7

SMILES

O=C(N(CCC1)[C@@H]1C(N)=O)[C@@H](NC([C@@H](NC2=O)CC(N2C)=O)=O)CC3=CN=CN3.CC(O)=O

CAS Number

1549593-23-8

Target & IC50

Thyrotropin-releasing hormone receptor: ic50 910nM

Product Categories/Family for Taltirelin acetate, inhibitor

Endocrinology/Hormones; Thyroid hormone receptor(THR)

Product References and Citations for Taltirelin acetate, inhibitor

Thirunarayanan N, et al. Taltirelin is a superagonist at the human thyrotropin-releasing hormone receptor. Front Endocrinol (Lausanne). 2012 Oct 9;3:120.

Other Notes

Small volumes of Taltirelin acetate, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Taltirelin acetate purchase

MBS5753999 is an inhibitor targeting Taltirelin acetate.