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TBOPP Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5754017

TBOPP is a selective DOCK1 inhibitor (IC50 : 8.4uM), with anti-tumor activity for broader types of tumors. More details

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Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
TBOPP, Inhibitor
Full Product Name
TBOPP
Product Gene Name
TBOPP, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
490.49
Solubility
DMSO: 120mg/mL (244.65mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C24H21F3N2O4S
SMILES
FC(F)(F)c1cccc(c1)-c1ccc(cc1)C(=O)Cn1cc(ccc1=O)S(=O)(=O)N1CCCC1
CAS Number
1996629-79-8
Target & IC50
DOCK1: ic50 8.4uM
DOCK1 DHR-2 domain: ic50 7.1uM (kd)
In Vitro
TBOPP treatment,suppressed cancer metastasis and growth in vivo in mice.

Structure of TBOPP, inhibitor

TBOPP Inhibitor – Cat# MBS5754017

Product References and Citations for TBOPP, inhibitor

Tajiri H, et al. Targeting Ras-Driven Cancer Cell Survival and Invasion through Selective Inhibition of DOCKCell Rep. 2017 May 2;19(5):969-980.

Other Notes

Small volumes of TBOPP, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for TBOPP purchase

MBS5754017 is an inhibitor targeting TBOPP.
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