Fanapanel Inhibitor

Name: Fanapanel Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5754163
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5754163

Fanapanel is a highly selective AMPA/kainate antagonist with little activity againstnMDA. It also has Ki values of 3.2nM, 100nM, and 8.5uM against quisqualate, kainate, andnMDA, respectively. More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Fanapanel, Inhibitor

Full Product Name

Fanapanel

Product Synonym Names

ZK200775; MPQX

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

409.25

Solubility

DMSO: 1.25mg/mL (3.05mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)

Formula

C14H15F3N3O6P

SMILES

O=C(N1CP(O)(O)=O)C(NC(C1=C2)=CC(C(F)(F)F)=C2N3CCOCC3)=O

CAS Number

161605-73-8

Target & IC50

AMPAR

Product Categories/Family for Fanapanel, inhibitor

Membrane Transporter/Ion Channel; Neuronal Signaling

Product References and Citations for Fanapanel, inhibitor

Turski L, et al. ZK200775: a phosphonate quinoxalinedione AMPA antagonist for neuroprotection in stroke and trauma. Proc Natl Acad Sci U S A. 1998 Sep 1;95(18):10960-5.
Kosowski AR, et al. Nicotine-induced dopamine release in the nucleus accumbens is inhibited by the novel AMPA antagonist ZK200775 and thenMDA antagonist CGP39551. Psychopharmacology (Berl). 2004 Aug;175(1):114-23.

Other Notes

Small volumes of Fanapanel, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Fanapanel purchase

MBS5754163 is an inhibitor targeting Fanapanel.