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(+)-Ketoconazole Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5754211

(+)-Ketoconazole is an agent of imidazole anti-fungal, and is an inhibitor of CYP3A4. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Product Name
(+)-Ketoconazole, Inhibitor
Full Product Name
(+)-Ketoconazole
Product Synonym Names
(+)-Ketoconazol; (+)-R 41400
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
531.43
Solubility
DMSO: 33.33mg/mL (62.72mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C26H28Cl2N4O4
SMILES
ClC(C=C1)=CC(Cl)=C1[C@@]2(CN3C=CN=C3)OC[C@H](COC4=CC=C(N5CCN(C(C)=O)CC5)C=C4)O2
CAS Number
142128-59-4
Target & IC50
Others

Structure of (+)-Ketoconazole, inhibitor

(+)-Ketoconazole Inhibitor – Cat# MBS5754211

Product References and Citations for (+)-Ketoconazole, inhibitor

Eil C. Ketoconazole binds to the human androgen receptor. Horm Metab Res. 1992 Aug;24(8):367-70.
Eil C. Ketoconazole binds to the human androgen receptor. Horm Metab Res. 1992 Aug;24(8):367-70.
Seif El-Din SH, et al. Effect of ketoconazole, a cytochrome P450 inhibitor, on the efficacy of quinine and halofantrine against Schistosoma mansoni in mice. Korean J Parasitol. 2013 Apr;51(2):165-75.
Seif El-Din SH, et al. Effect of ketoconazole, a cytochrome P450 inhibitor, on the efficacy of quinine and halofantrine against Schistosoma mansoni in mice. Korean J Parasitol. 2013 Apr;51(2):165-75.

Other Notes

Small volumes of (+)-Ketoconazole, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for (+)-Ketoconazole purchase

MBS5754211 is an inhibitor targeting (+)-Ketoconazole.
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