(+/-)-BAY-1251152 Inhibitor

Name: (+/-)-BAY-1251152 Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5754215
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5754215

(+/-)-BAY-1251152 is a racemic mixture of BAY-1251152. BAY-1251152 is highly selective inhibitor of PTEF/CDK9. More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

(+/-)-BAY-1251152, Inhibitor

Full Product Name

(+/-)-BAY-1251152

Product Gene Name

(+/-)-BAY-1251152, inhibitor

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

404.43

Solubility

DMSO: 50mg/mL (123.63mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)

Formula

C19H18F2N4O2S

SMILES

N=S(CC1=CC(NC2=NC=C(F)C(C3=CC=C(F)C=C3OC)=C2)=NC=C1)(C)=O

CAS Number

1610358-53-6

Target & IC50

Others

Product Categories/Family for (+/-)-BAY-1251152, inhibitor

Immunology/Inflammation; Nrf2; Others

Product References and Citations for (+/-)-BAY-1251152, inhibitor

Luecking, et al. Identification of potent and highly selective PTEFb inhibitor BAY 1251152 for the treatment,of cancer: from p.o. to i.v. application via scaffold hops [abstract]. In: Proceedings of the American Association for Cancer Research Annual Meeting 2017; 2017 Apr 1-5; Washington, DC. Philadelphia (PA): AACR; Cancer Res 2017;77(13 Suppl):Abstract nr 984. doi:10.1158/1538-7445. AM2017-984

Other Notes

Small volumes of (+/-)-BAY-1251152, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for (+/-)-BAY-1251152 purchase

MBS5754215 is an inhibitor targeting (+/-)-BAY-1251152.