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Apimostinel Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5754526

MBS5754526 is an inhibitor targeting Apimostinel. Apimostinel (NRX-1074; AGN-241660) is a partial agonist of nMDA receptor. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
Apimostinel, Inhibitor
Full Product Name
Apimostinel
Product Synonym Names
NRX-1074; AGN-241660
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
503.59
Solubility
DMSO: 155mg/mL (307.79mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C25H37N5O6
SMILES
C[C@@H](O)[C@@H](C(N)=O)NC([C@@]1(CC2=CC=CC=C2)N(C([C@H]3N(C([C@H]([C@H](O)C)N)=O)CCC3)=O)CCC1)=O
CAS Number
1421866-48-9
Target & IC50
Others
In Vitro
In preclinical models the two compounds both appear to be highly efficacious across a number of CNS disorders[1].

Structure of Apimostinel, inhibitor

Apimostinel Inhibitor – Cat# MBS5754526

Product References and Citations for Apimostinel, inhibitor

Naurex's First Orally Active Molecule, NRX-1074, Demonstrates Statistically Significant Improvement in Depression Scores within 24 Hours in Phase 2 Study for Major Depressive Disorder. January 28, 2015.
Naurex's First Orally Active Molecule, NRX-1074, Demonstrates Statistically Significant Improvement in Depression Scores within 24 Hours in Phase 2 Study for Major Depressive Disorder. January 28, 2015.

Other Notes

Small volumes of Apimostinel, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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