AZ-Dyrk1B-33 Inhibitor

Name: AZ-Dyrk1B-33 Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5754555
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5754555

AZ-Dyrk1B-33 is a potent and selective Dyrk1B kinase inhibitor. With an IC50 of 7nM[1]. More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

AZ-Dyrk1B-33, Inhibitor

Full Product Name

AZ-Dyrk1B-33

Product Gene Name

AZ-Dyrk1B-33, inhibitor

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

300.36

Solubility

<1mg/ml refers to the product slightly soluble or insoluble

Formula

C19H16N4

SMILES

CC1=NC=CC(C2=CN(CC3=CC=CC=C3)C4=C2C=CN=C4)=N1

CAS Number

1679330-37-0

Target & IC50

Dyrk1B: ic50 7nM

Product Categories/Family for AZ-Dyrk1B-33, inhibitor

Cell Cycle/Checkpoint; DYRK

Product References and Citations for AZ-Dyrk1B-33, inhibitor

Kettle JG, et al. Discovery and optimization of a novel series of Dyrk1B kinase inhibitors to explore a MEK resistance hypothesis. J Med Chem. 2015 Mar 26;58(6):2834-44.
Kettle JG, et al. Discovery and optimization of a novel series of Dyrk1B kinase inhibitors to explore a MEK resistance hypothesis. J Med Chem. 2015 Mar 26;58(6):2834-44.

Other Notes

Small volumes of AZ-Dyrk1B-33, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for AZ-Dyrk1B-33 purchase

MBS5754555 is an inhibitor targeting AZ-Dyrk1B-33.