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Bragsin1 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5754641

Bragsin1 is a potent and selective and noncompetitive ArfGEF BRAG2 inhibitor, inhibits Arf GTPase activation(IC50 : 3uM), and with anti-cancer activity. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
Bragsin1, Inhibitor
Full Product Name
Bragsin1
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
273.16
Solubility
DMSO: 62.5mg/mL (228.80mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C11H6F3NO4
SMILES
O=C1C=C(C(F)(F)F)OC2=CC=C(C)C([N+]([O-])=O)=C21
CAS Number
369631-68-5
Target & IC50
BRAG2: ic50 3uM

Structure of Bragsin1, inhibitor

Bragsin1 Inhibitor – Cat# MBS5754641

Product References and Citations for Bragsin1, inhibitor

Nawrotek A, et al. PH-domain-binding inhibitors of nucleotide exchange factor BRAG2 disrupt Arf GTPase signaling. Nat Chem Biol. 2019 Feb 1doi: 10.1038/s41589-019-0228-3.
Nawrotek A, et al. PH-domain-binding inhibitors of nucleotide exchange factor BRAG2 disrupt Arf GTPase signaling. Nat Chem Biol. 2019 Feb 11. doi: 10.1038/s41589-019-0228-3.

Other Notes

Small volumes of Bragsin1, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Bragsin1 purchase

MBS5754641 is an inhibitor targeting Bragsin1.
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