CGP36742 Inhibitor – CGP 36742

Name: CGP36742 Inhibitor; CGP 36742; MyBioSource
Brand: MyBioSource
SKU: MBS5754703
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5754703

CGP 36742 is a selective antagonist of the GABAB receptor that can penetrate the blood-brain barrier after peripheral administration (IC50: 32uM). It is useful in the treatment,of depression. More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

CGP 36742 (CGP36742), Inhibitor

Full Product Name

CGP 36742

Product Gene Name

CGP36742, inhibitor

Product Synonym Names

SGS-742

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

179.2

Solubility

<1mg/ml refers to the product slightly soluble or insoluble

Formula

C7H18NO2P

SMILES

O=P(CCCN)(O)CCCC

CAS Number

123690-78-8

Target & IC50

GABAB: ic50 32uM

Product Categories/Family for CGP36742, inhibitor

Membrane transporter/Ion channel; GABA Receptor; Neuroscience

Product References and Citations for CGP36742, inhibitor

Nowak G, et al. Antidepressant-like activity of CGP 36742 and CGP 51176, selective GABAB receptor antagonists, in rodents. Br J Pharmacol. 2006 Nov;149(5):581-90.
Nowak G, et al. Antidepressant-like activity of CGP 36742 and CGP 51176, selective GABAB receptor antagonists, in rodents. Br J Pharmacol. 2006 Nov;149(5):581-90.

Other Notes

Small volumes of CGP36742, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for CGP36742 purchase

MBS5754703 is an inhibitor targeting CGP36742. Also known as CGP 36742.