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CINPA1 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5754719

CINPA1 is a potent and specific inhibitor of the constitutive androstane receptor (CAR) that does not activate the PXR. CINPA1 reduces CAR-mediated transcription (IC50: ~70nM). More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
CINPA1, Inhibitor
Full Product Name
CINPA1
Product Gene Name
CINPA1, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
395.49
Solubility
DMSO: 250mg/mL (632.13mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C23H29N3O3
SMILES
CCN(CC)CC(N1C2=CC(NC(OCC)=O)=CC=C2CCC3=C1C=CC=C3)=O
CAS Number
102636-74-8
Target & IC50
CAR: ic50 ~70nM

Structure of CINPA1, inhibitor

CINPA1 Inhibitor – Cat# MBS5754719

Product References and Citations for CINPA1, inhibitor

Cherian MT, et al. CINPA1 is an inhibitor of constitutive androstane receptor that does not activate pregnane X receptor. Mol Pharmacol. 2015 May;87(5):878-89.
Cherian MT, et al. CINPA1 is an inhibitor of constitutive androstane receptor that does not activate pregnane X receptor. Mol Pharmacol. 2015 May;87(5):878-89.

Other Notes

Small volumes of CINPA1, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for CINPA1 purchase

MBS5754719 is an inhibitor targeting CINPA1.
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