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Dipraglurant Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5754792

MBS5754792 is an inhibitor targeting Dipraglurant. Dipraglurant is an antagonist of mGluR5 (IC50: 0.021uM). More details

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Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
Dipraglurant, Inhibitor
Full Product Name
Dipraglurant
Product Synonym Names
ADX48621
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
265.29
Solubility
DMSO: 40mg/mL (150.78mM)
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C16H12FN3
SMILES
FC1=CN2C(C=C1)=NC(CCC#CC3=NC=CC=C3)=C2
CAS Number
872363-17-2
Target & IC50
Others
In Vitro
Dipraglurant displayed in vivo activity in different anxiety models in rat50 and is currently in phase II for the treatment of dyskinesia in Parkinson's disease.

Structure of Dipraglurant, inhibitor

Dipraglurant Inhibitor – Cat# MBS5754792

Product References and Citations for Dipraglurant, inhibitor

The Synthesis and Use of Certain Pyridine Derivatives as Modulators of the G-protein Coupled Receptors mGlu5 and P2Y12
The Synthesis and Use of Certain Pyridine Derivatives as Modulators of the G-protein Coupled Receptors mGlu5 and P2Y12

Other Notes

Small volumes of Dipraglurant, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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