Esaxerenone Inhibitor

Name: Esaxerenone Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5754841
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5754841

Esaxerenone is a highly potent and selective non-steroidal antagonist of the mineralocorticoid receptor. More details

Please Inquire

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Esaxerenone, Inhibitor

Full Product Name

Esaxerenone

Product Synonym Names

CS-3150; XL-550

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

466.47

Solubility

DMSO: 125mg/mL (267.97mM)
(<1mg/ml refers to the product slightly soluble or insoluble)

Formula

C22H21F3N2O4S

SMILES

O=C(C1=CN(CCO)C(C2=CC=CC=C2C(F)(F)F)=C1C)NC3=CC=C(S(=O)(C)=O)C=C3

CAS Number

1632006-28-0

Target & IC50

Mineralocorticoid receptor

Product Categories/Family for Esaxerenone, inhibitor

Endocrinology/Hormones; Glucocorticoid Receptor

Product References and Citations for Esaxerenone, inhibitor

Yamada M, et al. Pharmacokinetics, distribution, and disposition of esaxerenone, a novel, highly potent and selective non-steroidal mineralocorticoid receptor antagonist, in rats and monkeys. Xenobiotica. 2017 Dec;47(12):1090-1103.
Yamada M, et al. Pharmacokinetics, distribution, and disposition of esaxerenone, a novel, highly potent and selective non-steroidal mineralocorticoid receptor antagonist, in rats and monkeys. Xenobiotica. 2017 Dec;47(12):1090-1103.

Other Notes

Small volumes of Esaxerenone, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Esaxerenone purchase

MBS5754841 is an inhibitor targeting Esaxerenone.