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Evatanepag Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5754848

Evatanepag is an agonist of EP2 receptor-selective prostaglandin E2 (PGE2). Which induces local bone formation (EC50: 0.3nM). More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
Evatanepag, Inhibitor
Full Product Name
Evatanepag
Product Synonym Names
CP-533536 free acid
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
468.57
Solubility
DMSO: 32mg/mL (68.29mM)
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C25H28N2O5S
SMILES
CC(C)(C)C(C=C1)=CC=C1CN(S(C2=CN=CC=C2)(=O)=O)CC3=CC(OCC(O)=O)=CC=C3
CAS Number
223488-57-1
Target & IC50
Others
In Vitro
Evatanepag (CP-533536) shows the ability to heal fractures when administered locally as a single dose in rat models of fracture healing s excellent in vitro potency and it also displays against EP2 and selectivity against a broad panel of other targets.

Structure of Evatanepag, inhibitor

Evatanepag Inhibitor – Cat# MBS5754848

Product References and Citations for Evatanepag, inhibitor

Cameron KO, et al. Discovery of CP-533536: an EP2 receptor selective prostaglandin E2 (PGE2) agonist that induces local bone formation. Bioorg Med Chem Lett. 2009 Apr 1;19(7):2075-8.
Cameron KO, et al. Discovery of CP-533536: an EP2 receptor selective prostaglandin E2 (PGE2) agonist that induces local bone formation. Bioorg Med Chem Lett. 2009 Apr 1;19(7):2075-8.

Other Notes

Small volumes of Evatanepag, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Evatanepag purchase

MBS5754848 is an inhibitor targeting Evatanepag.
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