Selisistat R-enantiomer Inhibitor

Name: Selisistat R-enantiomer Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5754852
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5754852

Selisistat R-enantiomer is much less active R-enantiomer of Selisistat (IC50 of > 100uM for SIRT1). More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Selisistat R-enantiomer, Inhibitor

Full Product Name

Selisistat R-enantiomer

Product Synonym Names

EX-527 (R-enantiomer)

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

248.71

Solubility

<1mg/ml refers to the product slightly soluble or insoluble

Formula

C13H13ClN2O

SMILES

O=C([C@H]1C(NC2=C3C=C(Cl)C=C2)=C3CCC1)N

CAS Number

848193-69-1

Target & IC50

SIRT1: ic50 >100uM

Product Categories/Family for Selisistat R-enantiomer, inhibitor

Chromatin/Epigenetic; Sirtuin; DNA Damage/DNA Repair

Product References and Citations for Selisistat R-enantiomer, inhibitor

Napper AD, et al. Discovery of indoles as potent and selective inhibitors of the deacetylase SIRTJ Med Chem. 2005 Dec 15;48(25):8045-54.
Napper AD, et al. Discovery of indoles as potent and selective inhibitors of the deacetylase SIRT1. J Med Chem. 2005 Dec 15;48(25):8045-54.

Other Notes

Small volumes of Selisistat R-enantiomer, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Selisistat R-enantiomer purchase

MBS5754852 is an inhibitor targeting Selisistat R-enantiomer.