Lidoflazine Inhibitor

Name: Lidoflazine Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5755101
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5755101

Lidoflazine is a high-affinity blocker of the HERG K+ channel and is an antianginal calcium channel blocker. It carries an obvious risk of QT interval prolongation and ventricular arrhythmia. More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Lidoflazine, Inhibitor

Full Product Name

Lidoflazine

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

491.62

Solubility

<1mg/ml refers to the product slightly soluble or insoluble

Formula

C30H35F2N3O

SMILES

O=C(NC1=C(C)C=CC=C1C)CN2CCN(CCCC(C3=CC=C(F)C=C3)C4=CC=C(F)C=C4)CC2

CAS Number

3416-26-0

Target & IC50

Ca2+

In Vitro

Lidoflazine inhibits effectively HERG current (IHERG). This recorded from HEK 293 cells stably expressing wild-type HERG (IC50: ~16nM).

Product Categories/Family for Lidoflazine, inhibitor

Membrane transporter/Ion channel; Calcium Channel

Product References and Citations for Lidoflazine, inhibitor

https://www.ncbi.nlm.nih.gov/pubmed/15135665
https://www.ncbi.nlm.nih.gov/pubmed/15135665

Other Notes

Small volumes of Lidoflazine, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Lidoflazine purchase

MBS5755101 is an inhibitor targeting Lidoflazine.