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LSZ-102 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5755120

LSZ-102 is an effective and orally bioavailable selective estrogen receptor degraded (IC50: 0.2nM). More details

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Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
LSZ-102, Inhibitor
Full Product Name
LSZ-102
Product Gene Name
LSZ-102, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
470.46
Solubility
DMSO: 100mg/mL (212.56mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C25H17F3O4S
SMILES
O=C(O)/C=C/C1=CC=C(OC2=C(C3=CC=C(F)C=C3C(F)(F)C)SC4=CC(O)=CC=C42)C=C1
CAS Number
2135600-76-7
Target & IC50
estrogen receptor

Structure of LSZ-102, inhibitor

LSZ-102 Inhibitor – Cat# MBS5755120

Product References and Citations for LSZ-102, inhibitor

Tria GS, et al. Discovery of LSZ102, a Potent, Orally Bioavailable Selective Estrogen Receptor Degrader (SERD) for the treatment,of Estrogen Receptor Positive Breast Cancer. J Med Chem. 2018 Apr 12;61(7):2837-2864.

Other Notes

Small volumes of LSZ-102, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for LSZ-102 purchase

MBS5755120 is an inhibitor targeting LSZ-102.
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