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LY2452473 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5755132

MBS5755132 is an inhibitor targeting LY2452473. LY2452473 is an orally bioavailable and selective androgen receptor modulator. More details

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Product Documentation
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Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
LY2452473, Inhibitor
Full Product Name
LY2452473
Product Gene Name
LY2452473, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
374.44
Solubility
DMSO: 62.5mg/mL (166.92mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C22H22N4O2
SMILES
O=C(N[C@@H]1CC(N(C2=C3C=C(C=C2)C#N)CC4=NC=CC=C4)=C3C1)OC(C)C
CAS Number
1029692-15-6
Target & IC50
Androgen receptor
In Vitro
LY2452473 is being developed for the treatment of disorders related to hypogonadism. LY2452473 is absorbed rapidly (time to reach maximum plasma concentration for both LY2452473 and total radioactivity is 2-3 h) and cleared slowly (plasma terminal t1/2 of 27 h for LY2452473 and 51 h for the total radioactivity).

Product Categories/Family for LY2452473, inhibitor

MAPK; Raf; Endocrinology/Hormones

Structure of LY2452473, inhibitor

LY2452473 Inhibitor – Cat# MBS5755132

Product References and Citations for LY2452473, inhibitor

Yi P, et al. Disposition and metabolism of LY2452473, a selective androgen receptor modulator, in humans. Drug Metab Dispos. 2012 Dec;40(12):2354-64.

Other Notes

Small volumes of LY2452473, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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