Propyl pyrazole triol Inhibitor

Name: Propyl pyrazole triol Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5755403
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5755403

Propyl pyrazole triol is a selective agonist of estrogen receptor alpha. The relative binding affinity of Propyl pyrazole triol for ERalpha (ERalpha: 49%) around 410 times higher compared with estrogen receptor beta (ERbeta: 0.12%). More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Propyl pyrazole triol, Inhibitor

Full Product Name

Propyl pyrazole triol

Product Synonym Names

PPT

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

386.44

Solubility

DMSO: 100mg/mL (258.77mM)
(<1mg/ml refers to the product slightly soluble or insoluble)

Formula

C24H22N2O3

SMILES

CCCC1=C(C2=CC=C(O)C=C2)N(C3=CC=C(O)C=C3)N=C1C4=CC=C(O)C=C4

CAS Number

263717-53-9

Target & IC50

Estrogen receptor alpha

Product References and Citations for Propyl pyrazole triol, inhibitor

Influence of cellular ERalpha/ERbeta ratio on the ERalpha-agonist induced proliferation of human T47D breast cancer cells.
Influence of cellular ERalpha/ERbeta ratio on the ERalpha-agonist induced proliferation of human T47D breast cancer cells.
Stauffer SR, et al. Pyrazole ligands: structure-affinity/activity relationships and estrogen receptor-alpha-selective agonists. J Med Chem. 2000 Dec 28;43(26):4934-47.
Stauffer SR, et al. Pyrazole ligands: structure-affinity/activity relationships and estrogen receptor-alpha-selective agonists. J Med Chem. 2000 Dec 28;43(26):4934-47.

Other Notes

Small volumes of Propyl pyrazole triol, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

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MBS5755403 is an inhibitor targeting Propyl pyrazole triol.

Propyl pyrazole triol Inhibitor

Product Overview

Structure of Propyl pyrazole triol, inhibitor

Related Product Information for Propyl pyrazole triol, inhibitor

Product References and Citations for Propyl pyrazole triol, inhibitor

Other Notes

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