Ritanserin Inhibitor

Name: Ritanserin Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5755462
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5755462

Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9nM). More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Ritanserin, Inhibitor

Full Product Name

Ritanserin

Product Synonym Names

R 55667

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

477.57

Solubility

DMSO: 25mg/mL (52.35mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)

Formula

C27H25F2N3OS

SMILES

CC1=C(C(N(C=CS2)C2=N1)=O)CCN(CC/3)CCC3=C(C4=CC=C(F)C=C4)\C5=CC=C(F)C=C5

CAS Number

87051-43-2

Target & IC50

5-HT2 receptor: ic50 0.9nM
H1 receptor: ic50 35nM
D2 receptor: ic50 70nM
alpha1 receptor: ic50 97nM
alpha2 receptor: ic50 150nM

Product Categories/Family for Ritanserin, inhibitor

GPCR/G Protein; 5-HT Receptor; Neuroscience

Product References and Citations for Ritanserin, inhibitor

Leysen JE, et al. Receptor-binding properties in vitro and in vivo of ritanserin: A very potent and long acting serotonin-S2 antagonist. Mol Pharmacol. 1985 Jun;27(6):600-11.
Leysen JE, et al. Receptor-binding properties in vitro and in vivo of ritanserin: A very potent and long acting serotonin-S2 antagonist. Mol Pharmacol. 1985 Jun;27(6):600-11.

Other Notes

Small volumes of Ritanserin, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Ritanserin purchase

MBS5755462 is an inhibitor targeting Ritanserin.