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Targapremir-210 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5755586

Targapremir-210 is an effective miR-210 inhibitor (IC50: 200nM in MDA-MB-231 cells). Targapremir-210 binds to the Dicer site of the miR-210 hairpin precursor. This interaction inhibits the production of mature miRNA. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
Targapremir-210, Inhibitor
Full Product Name
Targapremir-210
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
592.69
Solubility
DMSO: 250mg/mL (421.81mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C32H36N10O2
SMILES
O=C(NCCCN=[N+]=[N-])CCCOC1=CC=CC(C2=NC3=CC=C(C4=NC5=CC=C(N6CCN(C)CC6)C=C5N4)C=C3N2)=C1
CAS Number
1049722-30-6
Target & IC50
MDA-MB-231 cells: ic50 200nM

Structure of Targapremir-210, inhibitor

Targapremir-210 Inhibitor – Cat# MBS5755586

Product References and Citations for Targapremir-210, inhibitor

Costales MG, et al. Small Molecule Inhibition of microRNA-210 Reprograms an Oncogenic Hypoxic Circuit. J Am Chem Soc. 2017 Mar 8; 139(9):3446-3455.
Costales MG, et al. Small Molecule Inhibition of microRNA-210 Reprograms an Oncogenic Hypoxic Circuit. J Am Chem Soc. 2017 Mar 8; 139(9):3446-3455.

Other Notes

Small volumes of Targapremir-210, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Targapremir-210 purchase

MBS5755586 is an inhibitor targeting Targapremir-210.
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