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TUG-424 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5755664

TUG-424 significantly enhances glucose-stimulated insulin secretion at 100nM. TUG-424 is a potent and selective free fatty acid receptor 1 agonist (EC50: 32nM). More details

Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
TUG-424, Inhibitor
Full Product Name
TUG-424
Product Gene Name
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
264.32
Solubility
<1mg/ml refers to the product slightly soluble or insoluble
Formula
C18H16O2
SMILES
OC(CCC(C=C1)=CC=C1C#CC2=C(C)C=CC=C2)=O
CAS Number
1082058-99-8
Target & IC50
FFA1/GPR40: ic50 32nM (EC50)

Structure of TUG-424, inhibitor

TUG-424 Inhibitor – Cat# MBS5755664

Product References and Citations for TUG-424, inhibitor

Christiansen E, et al. Discovery of potent and selective agonists for the free fatty acid receptor 1 (FFA(1)/GPR40), a potential target for the treatment,of type II diabetes. J Med Chem. 2008 Nov 27;51(22):7061-4.

Other Notes

Small volumes of TUG-424, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for TUG-424 purchase

MBS5755664 is an inhibitor targeting TUG-424.
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