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UBP302 Inhibitor – UBP 302

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5755674

UBP 302 is an effective and selective GLUK5-subunit-containing kainate receptor antagonist (apparent Kd=402nM) and displays very little affinity on GluK2 kainate receptors. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
UBP 302 (UBP302), Inhibitor
Full Product Name
UBP 302
Product Gene Name
UBP302, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
333.3
Solubility
<1mg/ml refers to the product slightly soluble or insoluble
Formula
C15H15N3O6
SMILES
O=C(N(C=CC1=O)C[C@H](N)C(O)=O)N1CC2=C(C=CC=C2)C(O)=O
CAS Number
745055-91-8
Target & IC50
GLUK5: ic50 402nM (kd)

Structure of UBP302, inhibitor

UBP302 Inhibitor – Cat# MBS5755674

Product References and Citations for UBP302, inhibitor

Dolman NP, et al. Synthesis and pharmacology of willardiine derivatives acting as antagonists of kainate receptors. J Med Chem. 2005 Dec 1;48(24):7867-81.
Apland JP, et al. The limitations of diazepam as a treatment, for nerve agent-induced seizures and neuropathology in rats: comparison with UBP302. J Pharmacol Exp Ther. 2014 Nov;351(2):359-72.

Other Notes

Small volumes of UBP302, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for UBP302 purchase

MBS5755674 is an inhibitor targeting UBP302. Also known as UBP 302.
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