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Vercirnon Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5755694

Vercirnon is a selective and potent antagonist of CCR9 (IC50: 10nM). It is also used in the research of inflammatory bowel diseases. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
Vercirnon, Inhibitor
Full Product Name
Vercirnon
Product Synonym Names
GSK-1605786; CCX282-B; Traficet-EN
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
444.93
Solubility
DMSO: 25mg/mL (56.19mM)
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C22H21ClN2O4S
SMILES
O=S(C1=CC=C(C(C)(C)C)C=C1)(NC2=CC=C(Cl)C=C2C(C3=CC=[N+]([O-])C=C3)=O)=O
CAS Number
698394-73-9
Target & IC50
CCR9: ic50 10nM

Structure of Vercirnon, inhibitor

Vercirnon Inhibitor – Cat# MBS5755694

Product References and Citations for Vercirnon, inhibitor

Bekker P, et al. CCR9 Antagonists in the treatment,of Ulcerative Colitis. Mediators Inflamm. 2015;2015:628340.
Zhang J, et al. Biarylsulfonamide CCR9 inhibitors for inflammatory bowel disease. Bioorg Med Chem Lett. 2015 Sep 1;25(17):3661-4.

Other Notes

Small volumes of Vercirnon, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Vercirnon purchase

MBS5755694 is an inhibitor targeting Vercirnon.
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