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VU0529331 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5755706

VU0529331 is a modestly selective non-GIRK1-containing G protein-gated, inwardly-rectifying, potassium channel activator (EC50s: 5.1uM and 5.2uM for GIRK2 and GIRK1/2 in HEK293 cells, respectively). It is also effective on the GIRK4 homomeric channel. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
VU0529331, Inhibitor
Full Product Name
VU0529331
Product Gene Name
VU0529331, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
384.43
Solubility
<1mg/ml refers to the product slightly soluble or insoluble
Formula
C22H20N6O
SMILES
O=C(C1=NC=CN=C1)N2CC3=C(N4C=CC=C4)N(C5=CC(C)=C(C)C=C5)N=C3C2
CAS Number
1286725-49-2
Target & IC50
GIRK2: ic50 5.1uM (EC50)
GIRK1/2: ic50 5.2uM (EC50)

Structure of VU0529331, inhibitor

VU0529331 Inhibitor – Cat# MBS5755706

Product References and Citations for VU0529331, inhibitor

1. Kozek KA, et al. Discovery and Characterization of VU0529331, a Synthetic Small-Molecule Activator of Homomeric G Protein-Gated, Inwardly Rectifying, Potassium (GIRK) Channels. ACS Chem Neurosci. 2018 Sep 13.

Other Notes

Small volumes of VU0529331, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for VU0529331 purchase

MBS5755706 is an inhibitor targeting VU0529331.
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