WRG-28 Inhibitor

Name: WRG-28 Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5755714
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5755714

WRG-28 is a potent and selective, allosteric discoidin domain receptor 2 (ddr2) inhibitor(IC50 : 230nM) More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

WRG-28, Inhibitor

Full Product Name

WRG-28

Product Gene Name

WRG-28, inhibitor

Form/Format

Solid. Powder

Purity/Purification

97.84%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

410.44

Solubility

DMSO: 15mg/mL (36.55mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)

Formula

C21H18N2O5S

SMILES

CCNS(=O)(=O)c1ccc(COc2ccc3nc4ccc(=O)cc4oc3c2)cc1

CAS Number

1913291-02-7

Target & IC50

DDR2: ic50 230nM

Product Categories/Family for WRG-28, inhibitor

Tyrosine Kinase/Adaptors

Product References and Citations for WRG-28, inhibitor

Grither WR, et al. Inhibition of tumor-microenvironment interaction and tumor invasion by small-molecule allosteric inhibitor of DDR2 extracellular domain. Proc Natl Acad Sci U S A. 2018 Aug 14;115(33):E7786-E7794.

Other Notes

Small volumes of WRG-28, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for WRG-28 purchase

MBS5755714 is an inhibitor targeting WRG-28.