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PGlu-3-methyl-HIS-PRO-NH2 Inhibitor – TFA

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5756091

PGlu-3-methyl-His-Pro-NH2 TFA, enhances binding to pituitary TRH receptors and increases stimulation of thyroid-stimulating hormone (TSH) release from the pituitary. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
PGlu-3-methyl-His-Pro-NH2 TFA, Inhibitor
Full Product Name
PGlu-3-methyl-His-Pro-NH2 TFA
Product Gene Name
PGlu-3-methyl-His-Pro-NH2, inhibitor
Product Synonym Names
A-42872 TFA
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
490.43
Solubility
H2O: 250mg/mL (509.76mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C19H25F3N6O6
SMILES
CN1C(C[C@H](NC([C@@H](N2)CCC2=O)=O)C(N3[C@@H](CCC3)C(N)=O)=O)=CN=C1.OC(C(F)(F)F)=O
Target & IC50
Others
In Vitro
PGlu-3-methyl-His-Pro-NH2 TFA is more potent in eliciting behavioral effects as well as being more potent in the release of both growth hormone and thyroid stimulating hormone[1].

Structure of PGlu-3-methyl-His-Pro-NH2, inhibitor

PGlu-3-methyl-HIS-PRO-NH2 Inhibitor – Cat# MBS5756091

Product References and Citations for PGlu-3-methyl-His-Pro-NH2, inhibitor

Koskinen LO, et al. Cerebrovascular effects of the TRH analogues pGlu-3-methyl-His-Pro amide and pGlu-Glu-Pro amide: a comparison with TRH. Ups J Med Sci. 2000;105(1):73-83.
Koskinen LO, et al. Cerebrovascular effects of the TRH analogues pGlu-3-methyl-His-Pro amide and pGlu-Glu-Pro amide: a comparison with TRH. Ups J Med Sci. 2000;105(1):73-83.
Magnusson BM, et al. Biological effects after percutaneous absorption of thyrotropin-releasing hormone and its analogue M-TRH. Peptides. 2001 Jan;22(1):73-9.
Magnusson BM, et al. Biological effects after percutaneous absorption of thyrotropin-releasing hormone and its analogue M-TRH. Peptides. 2001 Jan;22(1):73-9.

Other Notes

Small volumes of PGlu-3-methyl-His-Pro-NH2, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for PGlu-3-methyl-His-Pro-NH2 purchase

MBS5756091 is an inhibitor targeting PGlu-3-methyl-His-Pro-NH2. Also known as PGlu-3-methyl-His-Pro-NH2 TFA.
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