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680C91 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5756784

MBS5756784 is an inhibitor targeting 680C91. 680C91 is a potent and selective inhibitor of TDO, and its Ki is 51nM. More details

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Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
680C91, Inhibitor
Full Product Name
680C91
Product Gene Name
680C91, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
238.26
Solubility
DMSO: 48mg/ml (201.46mM)
Ethanol: 25mg/ml (104.93mM)
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C15H11FN2
CAS Number
163239-22-3
Target & IC50
TDO: ic50 51nM (Ki)
Cell Research
Cell lines: rat liver cells. Concentrations: 0.1uM, 0.5uM, 2uM. Incubation Time: 0 min - 120 minutes. Method: The combined concentration of non-labelled L-tryptophan and the L-[ring-2-14C]-tryptophan used in the assays is 20uM and is added either with or without 68OC91 at time zero.

Product References and Citations for 680C91, inhibitor

M Salter, et al. Biochem Pharmacol. 1995 May 17;49(10):1435-42.
Sophie Imbeault, et al. Acta Neuropsychiatr. 2020 Feb;32(1):43-53.

Other Notes

Small volumes of 680C91, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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