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Protease-Activated Receptor-2, amide Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5758404

MBS5758404 is an inhibitor targeting Protease-Activated Receptor-2, amide. Protease-Activated Receptor-2, amide is an agonist of PAR2 (IC50 : 10.4 M) More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
Protease-Activated Receptor-2, amide, Inhibitor
Full Product Name
Protease-Activated Receptor-2, amide
Form/Format
Solid. Powder
Purity/Purification
100.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
614.78
Solubility
H2O: 33.33mg/mL (54.21mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C28H54N8O7
SMILES
CCC(C)C(NC(=O)C(CC(C)C)NC(=O)C(N)CO)C(=O)NCC(=O)NC(CCCCN)C(=O)NC(C(N)=O)C(C)C
CAS Number
190383-13-2
Target & IC50
PAR2: ic50 10.4 M

Product Categories/Family for Protease-Activated Receptor-2, amide, inhibitor

GPCR/G Protein

Structure of Protease-Activated Receptor-2, amide, inhibitor

Protease-Activated Receptor-2, amide Inhibitor – Cat# MBS5758404

Product References and Citations for Protease-Activated Receptor-2, amide, inhibitor

Kanke T, Ishiwata H, Kabeya M, et al. Binding of a highly potent protease-activated receptor-2 (PAR2) activating peptide, [~3H]2-furoyl-LIGRL-NH_2, to human PAR2[J]. British Journal of Pharmacology, 2005, 145(2):p.255-263.

Other Notes

Small volumes of Protease-Activated Receptor-2, amide, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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