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Taltirelin Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5758478

Taltirelin is at thyrotropin-releasing hormone receptor (TRH-R) superagonist (IC50 of 910nM and EC50 of 36nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release))[1]. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
Taltirelin, Inhibitor
Full Product Name
Taltirelin
Product Synonym Names
TA-0910
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
405.41
Solubility
DMSO: 30mg/mL (74mM)
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C17H23N7O5
SMILES
CN1C(=O)C[C@H](NC1=O)C(=O)N[C@@H](CC1=CN=CN1)C(=O)N1CCC[C@H]1C(N)=O
CAS Number
103300-74-9
Target & IC50
Thyrotropin-releasing hormone receptor

Structure of Taltirelin, inhibitor

Taltirelin Inhibitor – Cat# MBS5758478

Product References and Citations for Taltirelin, inhibitor

Dougherty J P, Wolff B S, Cullen M J, et al. Taltirelin alleviates fatigue-like behavior in mouse models of cancer-related fatigue.[J]. Pharmacological Research, 2017, 124:1-8.
Dougherty J P, Wolff B S, Cullen M J, et al. Taltirelin alleviates fatigue-like behavior in mouse models of cancer-related fatigue.[J]. Pharmacological Research, 2017, 124:1-8.
Thirunarayanan N, et al. Taltirelin is a superagonist at the human thyrotropin-releasing hormone receptor. Front Endocrinol (Lausanne). 2012 Oct 9;3:120.
Thirunarayanan N, et al. Taltirelin is a superagonist at the human thyrotropin-releasing hormone receptor. Front Endocrinol (Lausanne). 2012 Oct 9;3:120.

Other Notes

Small volumes of Taltirelin, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Taltirelin purchase

MBS5758478 is an inhibitor targeting Taltirelin.
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