diTFA Inhibitor – Protease-Activated Receptor-4

Name: diTFA Inhibitor; Protease-Activated Receptor-4; MyBioSource
Brand: MyBioSource
SKU: MBS5758621
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5758621

Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonist More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Protease-Activated Receptor-4 diTFA, Inhibitor

Full Product Name

Protease-Activated Receptor-4 diTFA (245443-52-1(free base))

Product Gene Name

diTFA, inhibitor

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

894.81

Solubility

<1mg/ml refers to the product slightly soluble or insoluble

Formula

C37H48F6N8O11

SMILES

OC(=O)C(F)(F)F.OC(=O)C(F)(F)F.NCCCC[C@H](NC(=O)CNC(=O)[C@@H]1CCCN1C(=O)[C@H](CC1=CC=C(O)C=C1)NC(=O)CN)C(=O)N[C@@H](CC1=CC=CC=C1)C(N)=O

Target & IC50

PAR-4

Product Categories/Family for diTFA, inhibitor

GPCR/G Protein; Protease-activated Receptor

Product References and Citations for diTFA, inhibitor

Huang S C. Proteinase-activated receptor-1 (PAR1) and PAR2 mediate relaxation of guinea pig internal anal sphincter[J]. Gastroenterology, 2014, 189(5):46-50.
Huang S C. Proteinase-activated receptor-1 (PAR1) and PAR2 mediate relaxation of guinea pig internal anal sphincter[J]. Gastroenterology, 2014, 189(5):46-50.
Moschonas I C, Kellici T F, Mavromoustakos T, et al. Molecular requirements involving the human platelet protease-activated receptor-4 mechanism of activation by peptide analogues of its tethered-ligand[J]. Platelets, 2017:1-10.
Moschonas I C, Kellici T F, Mavromoustakos T, et al. Molecular requirements involving the human platelet protease-activated receptor-4 mechanism of activation by peptide analogues of its tethered-ligand[J]. Platelets, 2017:1-10.

Other Notes

Small volumes of diTFA, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for diTFA purchase

MBS5758621 is an inhibitor targeting diTFA. Also known as Protease-Activated Receptor-4 diTFA (245443-52-1(free base)).