CZEN-002 Inhibitor

Name: CZEN-002 Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5758680
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5758680

CZEN-002 is amide stimulates melanocortin 1 receptor that results in the activation of adenylyl cyclase. More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

CZEN-002, Inhibitor

Full Product Name

CZEN-002

Product Gene Name

CZEN-002, inhibitor

Product Synonym Names

alpha-Melanocyte-Stimulating Hormone (MSH); amide

Form/Format

Solid. Powder

Purity/Purification

100.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

1664.88

Solubility

H2O: 50mg/mL (30.03mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)

Formula

C77H109N21O19S

SMILES

OC[C@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CO)NC(C)=O)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](Cc2cncn2)C(=O)N[C@@H](Cc3ccccc3)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc5cnc4ccccc45)C(=O)NCC(=O)N[C@@H](CCCCN)C(=O)N6CCC[C@H]6C(=O)N[C@H](C(N)=O)C(C)C

CAS Number

581-05-5

Target & IC50

Adenylyl cyclase

Product Categories/Family for CZEN-002, inhibitor

GPCR/G Protein

Product References and Citations for CZEN-002, inhibitor

Lu X Y, Barsh G S, Akil H, et al. Interaction between alpha-melanocyte-stimulating hormone and corticotropin-releasing hormone in the regulation of feeding and hypothalamo-pituitary-adrenal responses[J]. Journal of Neuroscience the Official Journal of the Society for Neuroscience, 2003, 23(21):7863.
Lu X Y, Barsh G S, Akil H, et al. Interaction between alpha-melanocyte-stimulating hormone and corticotropin-releasing hormone in the regulation of feeding and hypothalamo-pituitary-adrenal responses[J]. Journal of Neuroscience the Official Journal of the Society for Neuroscience, 2003, 23(21):7863.
Jo H, Choi M, Sim J, et al. Synthesis and Biological Evaluation of Caffeic Acid Derivatives as Potent Inhibitors of alpha-MSH-stimulated Melanogenesis[J]. Bioorganic & Medicinal Chemistry Letters, 2017:S0960894X17306133.
Jo H, Choi M, Sim J, et al. Synthesis and Biological Evaluation of Caffeic Acid Derivatives as Potent Inhibitors of alpha-MSH-stimulated Melanogenesis[J]. Bioorganic & Medicinal Chemistry Letters, 2017:S0960894X17306133.

Other Notes

Small volumes of CZEN-002, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for CZEN-002 purchase

MBS5758680 is an inhibitor targeting CZEN-002.