TBK1/IKKepsilon-IN-5 Inhibitor

Name: TBK1/IKKepsilon-IN-5 Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5758805
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5758805

TBK1/IKKepsilon-IN-5 is a dual TBK1 and IKKepsilon inhibitor(IC50 of 1nM and 5.6nM, respectively). More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

TBK1/IKKepsilon-IN-5, Inhibitor

Full Product Name

TBK1/IKKepsilon-IN-5

Product Gene Name

TBK1/IKKepsilon-IN-5, inhibitor

Form/Format

Solid. Powder

Purity/Purification

99.93%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

513.59

Solubility

DMSO: 7.81mg/mL (15.21mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)

Formula

C28H31N7O3

SMILES

N#Cc1cc(ccc1OC1CCOCC1)-c1ncnc(Nc2ccc(cc2)N2CCN(CC2)C2COC2)n1

CAS Number

1893397-65-3

Target & IC50

TBK1: ic50 1nM
IKKepsilon: ic50 5.6nM

Product Categories/Family for TBK1/IKKepsilon-IN-5, inhibitor

NF-kappab

Product References and Citations for TBK1/IKKepsilon-IN-5, inhibitor

Jenkins RW, et al. Ex Vivo Profiling of PD-1 Blockade Using Organotypic Tumor Spheroids. Cancer Discov. 2018 Feb;8(2):196-215.

Other Notes

Small volumes of TBK1/IKKepsilon-IN-5, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for TBK1/IKKepsilon-IN-5 purchase

MBS5758805 is an inhibitor targeting TBK1/IKKepsilon-IN-5.