Derenofylline Inhibitor

Name: Derenofylline Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5759119
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5759119

Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1nM) More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Derenofylline, Inhibitor

Full Product Name

Derenofylline

Form/Format

Solid. Powder

Purity/Purification

99.84%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

308.38

Solubility

<1mg/ml refers to the product slightly soluble or insoluble

Formula

C18H20N4O

SMILES

O[C@H]1CC[C@@H](CC1)Nc1nc(nc2[nH]ccc12)-c1ccccc1

CAS Number

251945-92-3

Target & IC50

adenosine A1 receptor: ic50 1nM (Ki)

Product Categories/Family for Derenofylline, inhibitor

GPCR/G Protein; Adenosine Receptor

Product References and Citations for Derenofylline, inhibitor

Kalk P, et al. The adenosine A1 receptor antagonist SLV320 reduces myocardial fibrosis in rats with 5/6 nephrectomy without affecting blood pressure. Br J Pharmacol. 2007 Aug;151(7):1025-32.

Other Notes

Small volumes of Derenofylline, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Derenofylline purchase

MBS5759119 is an inhibitor targeting Derenofylline.