Encequidar Inhibitor

MBS5759225 is an inhibitor targeting Encequidar. Encequidar is a potent and selective P-glycoprotein inhibitor.

Bauer F, et al. Interaction of HM30181 with P-glycoprotein at the murine blood-brain barrier assessed with positron emission tomography. Eur J Pharmacol. 2012 Dec 5;696(1-3):18-27.
Bauer F, et al. Interaction of HM30181 with P-glycoprotein at the murine blood-brain barrier assessed with positron emission tomography. Eur J Pharmacol. 2012 Dec 5;696(1-3):18-27.
Jin Cheul Kim, Kyeong Soo Kim, Dong Shik Kim,et al.Effect of HM30181 Mesylate Salt-Loaded Microcapsules on the Oral Absorption of Paclitaxel as a Novel P-glycoprotein Inhibitor. Int J Pharm. 2016 Jun 15;506(1-2):93-101.
Jin Cheul Kim, Kyeong Soo Kim, Dong Shik Kim,et al.Effect of HM30181 Mesylate Salt-Loaded Microcapsules on the Oral Absorption of Paclitaxel as a Novel P-glycoprotein Inhibitor. Int J Pharm. 2016 Jun 15;506(1-2):93-101.

Small volumes of Encequidar, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.