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Ripretinib Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5759275

MBS5759275 is an inhibitor targeting Ripretinib. Ripretinib is an orally bioavailable inhibitor of KIT and PDGFRA. More details

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Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
Ripretinib, Inhibitor
Full Product Name
Ripretinib
Product Synonym Names
DCC-2618
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
510.36
Solubility
DMSO: 40mg/mL (78.38mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C24H21BrFN5O2
SMILES
CCn1c2cc(NC)ncc2cc(-c2cc(NC(=O)Nc3ccccc3)c(F)cc2Br)c1=O
CAS Number
1442472-39-0
Target & IC50
Kit
PDGFR

Product Categories/Family for Ripretinib, inhibitor

Tyrosine Kinase/Adaptors; Angiogenesis

Structure of Ripretinib, inhibitor

Ripretinib Inhibitor – Cat# MBS5759275

Product References and Citations for Ripretinib, inhibitor

Schneeweiss M, et al. The KIT and PDGFRA switch-control inhibitor DCC-2618 blocks growth and survival of multiple neoplastic cell types in advanced mastocytosis. Haematologica. 2018 May;103(5):799-809.
Schneeweiss M, et al. The KIT and PDGFRA switch-control inhibitor DCC-2618 blocks growth and survival of multiple neoplastic cell types in advanced mastocytosis. Haematologica. 2018 May;103(5):799-809.

Other Notes

Small volumes of Ripretinib, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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