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BAY-545 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5759304

MBS5759304 is an inhibitor targeting BAY-545. BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59nM). More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
BAY-545, Inhibitor
Full Product Name
BAY-545
Product Gene Name
BAY-545, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
433.45
Solubility
DMSO: 145mg/mL (334.53mM)
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C18H22F3N3O4S
SMILES
CCn1c(=O)n(CCC(F)(F)F)c2sc(C(=O)N3CCC(O)CC3)c(C)c2c1=O
CAS Number
1699717-32-2
Target & IC50
A2B adenosine receptor: ic50 59nM
A2B adenosine receptor: ic50 59nM
Human A2B adenosine receptor: ic50 66nM
Mouse A2B adenosine receptor: ic50 400nM
Rat A2B adenosine receptor: ic50 280nM
Human A1 adenosine receptor: ic50 1300nM
Human A2A adenosine receptor: ic50 820nM
Mouse A2A adenosine receptor: ic50 470nM
Rat A2A adenosine receptor: ic50 750nM

Product Categories/Family for BAY-545, inhibitor

GPCR/G Protein

Structure of BAY-545, inhibitor

BAY-545 Inhibitor – Cat# MBS5759304

Product References and Citations for BAY-545, inhibitor

Harter M, et al. Novel non-xanthine antagonist of the A2B adenosine receptor: From HTS hit to lead structure. Eur J Med Chem.

Other Notes

Small volumes of BAY-545, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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