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Spastazoline Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5759305

Spastazoline is a potent and selective inhibitor of spastin(Human spastin with IC50 of 99nM). More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
Spastazoline, Inhibitor
Full Product Name
Spastazoline
Form/Format
Solid. Powder
Purity/Purification
100.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
382.51
Solubility
DMSO: 95mg/mL (248.36mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C20H30N8
SMILES
CC(C)[C@@H]1CN(CCN1)c1nc(Nc2cc([nH]n2)C(C)(C)C)c2cc[nH]c2n1
CAS Number
2351882-11-4
Target & IC50
Human spastin: ic50 99nM
spastin: ic50 99nM

Structure of Spastazoline, inhibitor

Spastazoline Inhibitor – Cat# MBS5759305

Product References and Citations for Spastazoline, inhibitor

Cupido T, et al. Designing a chemical inhibitor for the AAA protein spastin using active site mutations. Nat Chem Biol. 2019 Feb
Cupido T, et al. Designing a chemical inhibitor for the AAA protein spastin using active site mutations. Nat Chem Biol. 2019 Feb
Pisa R, Cupido T, Steinman J B, et al. Analyzing Resistance to Design Selective Chemical Inhibitors for AAA Proteins[J].
Pisa R, Cupido T, Steinman J B, et al. Analyzing Resistance to Design Selective Chemical Inhibitors for AAA Proteins[J].

Other Notes

Small volumes of Spastazoline, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Spastazoline purchase

MBS5759305 is an inhibitor targeting Spastazoline.
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