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PACAP Inhibitor – TFA

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5763383

PACAP (1-27), human, ovine, rat TFA (PACAP 1-27 TFA) is an N-terminal fragment of pacap-38 and an effective PACAP receptor antagonist. The IC50s for rat PAC1, rat VPAC1 and human VPAC2 are 3nm, 2nm and 5nm respectively. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
PACAP TFA, Inhibitor
Full Product Name
PACAP (1-27), human, ovine, rat TFA
Product Gene Name
PACAP, inhibitor
Product Synonym Names
PACAP 1-27 TFA
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
3261.68
Solubility
H2O: 100mg/mL (30.66mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C144H225F3N40O41S
Target & IC50
rat PAC1: ic50 3nM
rat VPAC1: ic50 2nM
human VPAC2: ic50 5nM

Product References and Citations for PACAP, inhibitor

Gourlet P, et al. Fragments of pituitary adenylate cyclase activating polypeptide discriminate between type I and II recombinant receptors. Eur J Pharmacol. 1995 Dec 4;287(1):7-11.
Schafer H, et al. Structural motifs of pituitary adenylate cyclase-activating polypeptide (PACAP) defining PAC1-receptor selectivity. Regul Pept. 1999 Feb 5;79(2-3):83-92.
Linden A, et al. Inhibition of bronchoconstriction by pituitary adenylate cyclase activating polypeptide (PACAP 1-27) in guinea-pigs in vivo. Br J Pharmacol. 1995 Jul;115(6):913-6.

Other Notes

Small volumes of PACAP, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for PACAP purchase

MBS5763383 is an inhibitor targeting PACAP. Also known as PACAP (1-27), human, ovine, rat TFA.
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