• Call +1.858.633.0165 or Fax +1.858.633.0166 or Contact Us

K-(D-1-NAL)-FwLL-NH2 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5763892

High affinity and potent ghrelin receptor inverse agonist (Ki values are 4.9 and 31nM in COS7 and HEK293T cells, respectively). Blocks ghrelin receptor-mediated Gq- and G13-dependent signaling pathways. More details

Please Inquire
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
K-(D-1-Nal)-FwLL-NH2, Inhibitor
Full Product Name
K-(D-1-Nal)-FwLL-NH2
Product Gene Name
K-(D-1-Nal)-FwLL-NH2, inhibitor
Product Synonym Names
K-(D-1-Nal)-FwLL-NH2
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
902.13
Solubility
Water: 2mg/mL
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C51H67N9O6
CAS Number
1394288-22-2

Product References and Citations for K-(D-1-Nal)-FwLL-NH2, inhibitor

Els et al (2012) An aromatic region to induce a switch between agonism and inverse agonism at the ghrelin receptor. J.Med.Chem. 55 7437 PMID:
Els et al (2012) An aromatic region to induce a switch between agonism and inverse agonism at the ghrelin receptor. J.Med.Chem. 55 7437 PMID:
M'Kadmi et al (2015) Agonism, antagonism, and inverse agonism bias at the ghrelin receptor signaling. J. Biol.Chem. 290 27021 PMID:
M'Kadmi et al (2015) Agonism, antagonism, and inverse agonism bias at the ghrelin receptor signaling. J. Biol.Chem. 290 27021 PMID:

Other Notes

Small volumes of K-(D-1-Nal)-FwLL-NH2, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for K-(D-1-Nal)-FwLL-NH2 purchase

MBS5763892 is an inhibitor targeting K-(D-1-Nal)-FwLL-NH2.
Request a Quote

Please fill out the form below and our representative will get back to you shortly.

MBS000000
Contact Us

Please fill out the form below and our representative will get back to you shortly.

MBS000000