AZ3451 Inhibitor

Name: AZ3451 Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5764270
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5764270

AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23nM). More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

AZ3451, Inhibitor

Full Product Name

AZ3451

Product Gene Name

AZ3451, inhibitor

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

571.46

Solubility

DMSO: 80mg/mL (140mM)
Water: Insoluble
(<1mg/ml refers to the product slightly soluble or insoluble)

Formula

C30H27BrN4O3

SMILES

C[C@@H](C1CCCCC1)n1c(-c(cc2OCOc2c2)c2Br)nc2c1ccc(C(Nc(cc1)ccc1C#N)=O)c2

CAS Number

2100284-59-9

Product Categories/Family for AZ3451, inhibitor

GPCR/G Protein; Protease-activated Receptor

Product References and Citations for AZ3451, inhibitor

Cheng RKY, et al. Structural insight into allosteric modulation of protease-activated receptor 2. Nature. 2017 May 4;545(7652):112-115.

Other Notes

Small volumes of AZ3451, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for AZ3451 purchase

MBS5764270 is an inhibitor targeting AZ3451.