Nastorazepide Inhibitor

Name: Nastorazepide Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5764320
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5764320

Nastorazepide (Z-360) is a selective, orally available antagonist of gastrin/cholecystokinin 2 (CCK-2) receptor with potential antineoplastic activity. More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Nastorazepide, Inhibitor

Full Product Name

Nastorazepide

Product Synonym Names

Z-360

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

520.62

Solubility

DMSO: 30mg/mL (57.63mM)
(<1mg/ml refers to the product slightly soluble or insoluble)

Formula

C29H35N4O5

SMILES

O=C(O)C1=CC=CC(NC(N[C@]2C(N(CC(C(C)(C)C)=O)C3=CC=CC=C3N(C4CCCCC4)C2)=O)=O)=C1

CAS Number

209219-38-5

In Vitro

Z-360 significantly inhibits the growth of subcutaneous xenografts of human pancreatic tumor cells in mice, and that Z-360 combined with gemcitabine prolonged survival in a pancreatic carcinoma orthotopic xenograft mice.

Product Categories/Family for Nastorazepide, inhibitor

GPCR/G Protein; cholecystokinin

Product References and Citations for Nastorazepide, inhibitor

Kato H, et al. CCK-2/gastrin receptor signaling pathway is significant for gemcitabine-induced gene expression of VEGF in pancreatic carcinoma cells. Life Sci. 2011 Oct 24;89(17-18):603-8.

Other Notes

Small volumes of Nastorazepide, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Nastorazepide purchase

MBS5764320 is an inhibitor targeting Nastorazepide.