GR79236 Inhibitor – Gr 79236

Name: GR79236 Inhibitor; Gr 79236; MyBioSource
Brand: MyBioSource
SKU: MBS5764392
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5764392

GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1nM) that has analgesic and anti-inflammatory actions. More details

Please Inquire

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

GR 79236 (GR79236), Inhibitor

Full Product Name

GR 79236

Product Gene Name

GR79236, inhibitor

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

351.36

Solubility

Water: 98mg/mL (278.92mM)
(<1mg/ml refers to the product slightly soluble or insoluble)

Formula

C15H17N5O5

SMILES

O[C@]1[C@@H](N2C3=NC=NC(N[C@@H](CCC4)[C@]4O)=C3N=C2)O[C@](CO)[C@]1O

CAS Number

124555-18-6

In Vitro

GR79236 has been shown to have antinociceptive and anti-inflammatory properties in animal models. GR79236 inhibits the release of CGRP evoked by superior sagittal sinus (SSS) stimulation in the cat and inhibits trigeminal nucleus firing in the cat and rat. GR79236X has acute, short-term analgesic efficacy.

Product Categories/Family for GR79236, inhibitor

GPCR/G Protein; Adenosine Receptor

Product References and Citations for GR79236, inhibitor

Sneyd JR, et al. Multicentre evaluation of the adenosine agonist GR79236X in patients with dental pain after third molar extraction. Br J Anaesth. 2007 May;98(5):672-676.
Sneyd JR, et al. Multicentre evaluation of the adenosine agonist GR79236X in patients with dental pain after third molar extraction. Br J Anaesth. 2007 May;98(5):672-676.
Arulmani U, et al. Lack of effect of the adenosine A1 receptor agonist, GR79236, on capsaicin-induced CGRP release in anaesthetized pigs. Cephalalgia. 2005 Nov;25(11):1082-90.
Arulmani U, et al. Lack of effect of the adenosine A1 receptor agonist, GR79236, on capsaicin-induced CGRP release in anaesthetized pigs. Cephalalgia. 2005 Nov;25(11):1082-90.

Other Notes

Small volumes of GR79236, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GR79236 purchase

MBS5764392 is an inhibitor targeting GR79236. Also known as GR 79236.