MSC2530818 Inhibitor

Name: MSC2530818 Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5764516
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5764516

MSC2530818 is an effective, selective and orally available CDK8 inhibitor (IC50: 2.6nM). More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

MSC2530818, Inhibitor

Full Product Name

MSC2530818

Product Gene Name

MSC2530818, inhibitor

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

340.81

Solubility

DMSO: 120mg/mL (352.1mM)
(<1mg/ml refers to the product slightly soluble or insoluble)

Formula

C18H17ClN4O

SMILES

Cc1[nH]nc2ncc(cc12)C(=O)N1CCC[C@H]1c1ccc(Cl)cc1

CAS Number

1883423-59-3

Product Categories/Family for MSC2530818, inhibitor

Cell Cycle/Checkpoint; CDK

Product References and Citations for MSC2530818, inhibitor

Czodrowski P, et al. Structure-Based Optimization of Potent, Selective, and Orally Bioavailable CDK8 Inhibitors Discovered by High-Throughput Screening. J Med Chem. 2016 Oct 27;59(20):9337-9349.

Other Notes

Small volumes of MSC2530818, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for MSC2530818 purchase

MBS5764516 is an inhibitor targeting MSC2530818.