Cenicriviroc (TAK-652)

Name: Cenicriviroc (TAK-652); MyBioSource
Brand: MyBioSource
SKU: MBS8400467
Price: 205 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS8400467

Cenicriviroc is a potent inhibitor of C-C chemokine receptors CCR5 and CCR2. It is an orally bioavailable derivative of TAK-779 with potent anti-HIV-1 activity. It blocks the binding of MIP-1alpha and MIP-1beta to CCR5 with an IC50 of 2.3nM. It inhibits the… More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Product Name

Cenicriviroc, Biochemical

Full Product Name

Cenicriviroc

Product Synonym Names

TAK-652; TBR-652; (5E)-8-[4-(2-butoxyethoxy)phenyl]-1-(2-methylpropyl)-N-[4-[(S)-(3-propylimidazol-4-yl)methylsulfinyl]phenyl]-3, 4-dihydro-2H-1-benzazocine-5-carboxamide; (S, E)-8-(4-(2-butoxyethoxy)phenyl)-1-isobutyl-N-(4-(((1-propyl-1H-imidazol-5-yl)methyl)sulfinyl)phenyl)-1, 2, 3, 4-tetrahydrobenzo[b]azocine-5-carboxamide

Form/Format

Yellow Solid

Purity/Purification

>=98%

Specificity

A potent inhibitor of CCR5 and CCR2

Preparation and Storage

Store at -20 degree C
Do not take internally. Wear gloves and mask when handling the product! Avoid contact by all modes of exposure.
Shipping: Gel Pack
Shelf Life: Est.~36months
Country of Origin: USA

Molecular Weight

696.94

Solubilities

~5mg/ml in ethanol; ~20mg/ml in DMSO and DMF

Molecular Formula

C??H??N?O?S

InChi

InChI=1S/C41H52N4O4S/c1-5-7-22-48-23-24-49-38-15-10-32(11-16-38)33-12-19-40-35(25-33)26-34(9-8-21-44(40)28-31(3)4)41(46)43-36-13-17-39(18-14-36)50(47)29-37-27-42-30-45(37)20-6-2/h10-19; 25-27; 30-31H; 5-9; 20-24; 28-29H2; 1-4H3; (H; 43; 46)/b34-26+/t50-/m0/s1

InChi Key

PNDKCRDVVKJPKG-WHERJAGFSA-N

SMILES

CCCCOCCOC1=CC=C(C=C1)C2=CC3=C(C=C2)N(CCCC(=C3)C(=O)NC4=CC=C(C=C4)S(=O)CC5=CN=CN5CCC)CC(C)C

CAS Number

497223-25-3

MDL Number

MFCD28502076

PubChem CID

11285792

Product Categories/Family for Cenicriviroc biochemical

Web Categories; Biochemicals; Biochemicals (A-Z); Antiviral Agents

Product References and Citations for Cenicriviroc biochemical

https://pubchem.ncbi.nlm.nih.gov/compound/11285792

Other Notes

Small volumes of Cenicriviroc biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Cenicriviroc purchase

MBS8400467 is a biochemical targeting Cenicriviroc.