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OTX015

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS842260

Background: OTX015 is a potent inhibitor of BRD2, BRD3, and BRD4 (EC??s = 10-19 nM). It displays antiproliferative effects at a sub-micromolar range in vitro in a wide range of solid tumor types and leukemias, downregulating c-Myc expression and inducing… More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Product Name
OTX015, Biochemical
Full Product Name
OTX015
Product Gene Name
OTX015 biochemical
Product Synonym Names
(6S)-4-(4-chlorophenyl)-N-(4-hydroxyphenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide; HY-15743
Form/Format
Appearance: Crystaline solid
Purity/Purification
>=98%
Preparation and Storage
At -20 degree C
Shelf Life: 36 months
Molecular Weight
492
CAS Number
202590-98-5
Structure Available?
Yes
Salt Form
No
Cell-Permeable?
Yes
PubChem CID
9936746
Solubility/Reconstitution Instructions
DMSO (~25 mg/ml) or EtOH (~ 25 mg/ml)
SMILES
 CC1=C(SC2=C1C(=NC(C3=NN=C(N32)C)CC(=O)NC4=CC=C(C=C4)O)C5=CC=C(C=C5)Cl)C
InChi
nChI=1S/C25H22ClN5O2S/c1-13-14(2)34-25-22(13)23(16-4-6-17(26)7-5-16)28-20(24-30-29-15(3)31(24)25)12-21(33)27-18-8-10-19(32)11-9-18/h4-11,20,32H,12H2,1-3H3,(H,27,33)/t20-/m0/s1
InChi Key
GNMUEVRJHCWKTO-FQEVSTJZSA-N
Handling
Protect from air and light

Product Categories/Family for OTX015 biochemical

Enzyme Inhibitors; Bromodomain InhibitorsBiochemicals; Enzyme Inhibitors; Bromodomain InhibitorsEpigenetics; Reader Domains; Bromodomains; Bromodomain InhibitorsBiochemicals; Biochemicals (A-Z)

Structure of OTX015 biochemical

OTX015 Biochemical – Cat# MBS842260

Other Notes

Small volumes of OTX015 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for OTX015 purchase

MBS842260 is a biochemical targeting OTX015.
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