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HTH-01-015

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS842629

Background: HTH-01-015 is a potent and selective inhibitor of NUAK1 kinase (IC?? =100 nM); only weakly inhibits NUAK2 (IC?? of >10 muM) and does not significantly inhibit the activity of 139 other kinases that were tested including ten AMPK family members. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Product Name
HTH-01-015, Biochemical
Full Product Name
HTH-01-015
Product Synonym Names
4,5,13-trimethyl-2-((1-(piperidin-4-yl)-1H-pyrazol-4-yl)amino)-5H-naphtho[2,3-e]pyrimido[5,4-b][1,4]diazepin-6(13H)-one
Form/Format
Appearance: Crystalline solid
Purity/Purification
>=98% by HPLC
Preparation and Storage
At -20 degree C
Shelf Life: 36 months
Molecular Weight
468.55
CAS Number
1613724-42-7 
Structure Available?
Yes
Salt Form
No
Cell-Permeable?
Yes
PubChem CID
78357766
Solubility/Reconstitution Instructions
DMSO
SMILES
CC1=C2C(=NC(=N1)NC3=CN(N=C3)C4CCNCC4)N(C5=CC6=CC=CC=C6C=C5C(=O)N2C)C
InChi
nChI=1S/C26H28N8O/c1-16-23-24(31-26(29-16)30-19-14-28-34(15-19)20-8-10-27-11-9-20)32(2)22-13-18-7-5-4-6-17(18)12-21(22)25(35)33(23)3/h4-7,12-15,20,27H,8-11H2,1-3H3,(H,29,30,31)
InChi Key
CHSDJDLAKKAWCI-UHFFFAOYSA-N
Handling
Protect from air and light

Product Categories/Family for HTH-01-015 biochemical

Enzyme Inhibitors; Protein Kinase Inhibitors; Other Protein Kinase InhibitorsEnzyme Inhibitors; Enzyme Inhibitors (A-Z) Biochemicals; Enzyme Inhibitors; Protein Kinase Inhibitors; Other Protein Kinase InhibitorsBiochemicals; Enzyme Inhibitors; Enzyme Inhi

Structure of HTH-01-015 biochemical

HTH-01-015 Biochemical – Cat# MBS842629

Other Notes

Small volumes of HTH-01-015 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for HTH-01-015 purchase

MBS842629 is a biochemical targeting HTH-01-015.
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