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I-BET762

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS842743

Background: I-BET762 (GSK525762) is a highly potent, selective and cell-permeable inhibitor of the bromodomain and extra terminal (BET) family protein BRD4 (IC?? of ~35 nM). It inhibits myeloma cell proliferation and suppresses the production of… More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Product Name
I-BET762, Biochemical
Full Product Name
I-BET762
Product Gene Name
I-BET762 biochemical
Product Synonym Names
(4S)-6-(4-Chlorophenyl)-N-ethyl-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine-4-acetamide; GSK525762
Form/Format
Appearance: Off-white solid
Purity/Purification
>98% by HPLC
Preparation and Storage
At -20 degree C
Shelf Life: 36 months
Molecular Weight
423.9
CAS Number
1260907-17-2
Structure Available?
Y
Salt Form
No
Cell-Permeable?
Yes
PubChem CID
46943432
Solubility/Reconstitution Instructions
DMSO or EtOH
SMILES
 CCNC(=O)CC1C2=NN=C(N2C3=C(C=C(C=C3)OC)C(=N1)C4=CC=C(C=C4)Cl)C
InChi
nChI=1S/C22H22ClN5O2/c1-4-24-20(29)12-18-22-27-26-13(2)28(22)19-10-9-16(30-3)11-17(19)21(25-18)14-5-7-15(23)8-6-14/h5-11,18H,4,12H2,1-3H3,(H,24,29)/t18-/m0/s1
InChi Key
AAAQFGUYHFJNHI-SFHVURJKSA-N
Handling
Protect from air and light

Product Categories/Family for I-BET762 biochemical

Enzyme Inhibitors; Bromodomain InhibitorsBiochemicals; Enzyme Inhibitors; Bromodomain InhibitorsEpigenetics; Reader Domains; Bromodomains; Bromodomain InhibitorsEpigenetics; Epigenetic Modulators (A-Z) Biochemicals; Biochemicals (A-Z)

Structure of I-BET762 biochemical

I-BET762 Biochemical – Cat# MBS842743

Other Notes

Small volumes of I-BET762 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for I-BET762 purchase

MBS842743 is a biochemical targeting I-BET762.
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