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GSK-3787

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS842896

Background: GSK-3787 is a selective and irreversible antagonist of the peroxisome proliferator-activated receptor delta (PPARdelta) (plC?? = 6.6). It covalently binds to Cys 249 in the PPARdelta binding site. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Product Name
GSK-3787, Biochemical
Full Product Name
GSK-3787
Product Gene Name
GSK-3787 biochemical
Product Synonym Names
4-Chloro-N-(2-{[5-(trifluoromethyl)-2-pyridyl]sulfonyl}ethyl)benzamide
Form/Format
Appearance: White solid
Purity/Purification
>=98% by TLC
Preparation and Storage
At -20 degree C
Shelf Life: 36 months
Molecular Weight
392.78
CAS Number
188591-46-0
Structure Available?
Yes
Salt Form
No
Cell-Permeable?
Yes
MDL Number
MFCD00099612
PubChem CID
2800647
Solubility/Reconstitution Instructions
DMSO (~30 mg/ml)
SMILES
C1=CC(=CC=C1C(=O)NCCS(=O)(=O)C2=NC=C(C=C2)C(F)(F)F)Cl
InChi
InChI=1S/C15H12ClF3N2O3S/c16-12-4-1-10(2-5-12)14(22)20-7-8-25(23,24)13-6-3-11(9-21-13)15(17,18)19/h1-6,9H,7-8H2,(H,20,22)
InChi Key
JFUIMTGOQCQTPF-UHFFFAOYSA-N
Handling
Protect from light and air

Product Categories/Family for GSK-3787 biochemical

Enzyme Inhibitors; PPAR Antagonists and Biochemicals; Enzyme Inhibitors; PPAR Antagonists and Diabetes; Obesity & Metabolic Syndrome; Signaling Pathways in Diabetes and Obesity; PPAR Signaling; PPAR Antagonists and Biochemicals; Biochemicals (A-Z)

Structure of GSK-3787 biochemical

GSK-3787 Biochemical – Cat# MBS842896

Other Notes

Small volumes of GSK-3787 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GSK-3787 purchase

MBS842896 is a biochemical targeting GSK-3787.
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