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RGB-286638, free base

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS842956

Background: RGB-286638 is a potent and selective cyclin-dependent kinase (CDK) inhibitor with IC?? values of 1, 2, 3 and 44 nM for CDK9, CDK1, CDK2, and CDK4, respectively.  Less potent against cyclin H-CDK7 and cyclin D3-CDK6. It inhibits cell cycle… More details

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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Product Overview

Product Name
RGB-286638, Biochemical
Full Product Name
RGB-286638, free base
Product Gene Name
RGB-286638 biochemical
Product Synonym Names
1-[3-[4-[[4-(2-methoxyethyl)piperazin-1-yl]methyl]phenyl]-4-oxo-1H-indeno[1,2-c]pyrazol-5-yl]-3-morpholin-4-ylurea
Form/Format
Appearance: Crystalline solid
Purity/Purification
>=98% by HPLC
Preparation and Storage
At -20 degree C
Shelf Life: 36 months
Molecular Weight
545.63
CAS Number
784210-88-4 
Structure Available?
Yes
Salt Form
No
Cell-Permeable?
Yes
PubChem CID
11285002
Solubility/Reconstitution Instructions
DMSO
SMILES
COCCN1CCN(CC1)CC2=CC=C(C=C2)C3=NNC4=C3C(=O)C5=C4C=CC=C5NC(=O)NN6CCOCC6
InChi
InChI=1S/C29H35N7O4/c1-39-16-13-34-9-11-35(12-10-34)19-20-5-7-21(8-6-20)26-25-27(32-31-26)22-3-2-4-23(24(22)28(25)37)30-29(38)33-36-14-17-40-18-15-36/h2-8H,9-19H2,1H3,(H,31,32)(H2,30,33,38)
InChi Key
XLSYZSRXVVCHLS-UHFFFAOYSA-N
Handling
Protect from air and light

Product Categories/Family for RGB-286638 biochemical

Enzyme Inhibitors; Protein Kinase Inhibitors; CDK InhibitorsEnzyme Inhibitors; Enzyme Inhibitors (A-Z) Biochemicals; Enzyme Inhibitors; Protein Kinase Inhibitors; CDK InhibitorsBiochemicals; Enzyme Inhibitors; Enzyme Inhibitors (A-Z) Biochemicals; Biochem

Structure of RGB-286638 biochemical

RGB-286638, free base Biochemical – Cat# MBS842956

Other Notes

Small volumes of RGB-286638 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for RGB-286638 purchase

MBS842956 is a biochemical targeting RGB-286638. Also known as RGB-286638, free base.
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